Paracetamol in Horses (Equis) | Vetlexicon
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Paracetamol


Introduction

Name

  • Paracetamol.

Class of drug

  • Aniline analgesic.
  • Non-steroidal anti-inflammatory drug (NSAID).

Description

  • Stop administration of drug.
  • May administer activated charcoal is diagnosed rapidly (<1 h).
  • Supportive or symptomatic treatment, eg intravenous fluids.
  • May require other treatments such as N-acetycysteine (see below), blood transfusion.
  • Monitor liver and renal blood test parameters.

Uses

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Administration

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Pharmacokinetics

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Precautions

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Withdrawal Periods

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Adverse Reactions

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Further Reading

Publications

Refereed papers

  • Recent references from PubMed and VetMedResource.
  • West E et al (2011) Use of acetaminophen (paracetamol) as a short-term adjunctive analgesic in a laminitic pony. Vet Anaesthesia Analgesia 38 (5), 521-522 PubMed.
  • Neirinckx E et al (2010) Species comparison of oral bioavailability, first-pass metabolism and pharmacokinetics of acetaminophen. Res Vet Sci 89 (1), 113-119 PubMed.
  • Pickering G et al (2006) Analgesic effect of acetaminophen in humans: first evidence of a central serotonergic mechanism. Clin Pharmacol Therapeutics 79 (4), 371-378.
  • Greenblatt D J & Engelking L R (1988) Enterohepatic circulation of lorazepam and acetaminophen conjugates in ponies. J Pharmacol Exper Therapeutics 244 (2), 674-679 PubMed.